NPEdia

FSL0312

Structure
FSL0312
Synonyms
Origin
Chemically synthesized
Biological activities
β-adrenoreceptor antagonist
Mild intrinsic sympathomimetic activity
Therapeutic
Antiangina
Antiarrhythmic (class II)
Antihypertensive
Target
Selective β1-adrenergic receptors
Assay information
Effects on the activation of Adenylate cyclase from heart and liver induced by 1-isoproterenol (IC50 [μM]): Heart (9.0), Liver (838.9)
Isoprenaline-induced tachycardia and diastolic hypotension antagonize avtivity