NPEdia

FSL0739

Structure
FSL0739
Synonyms
Origin
Streptomyces niveus
Biological activities
Inhibition of DNA replication in bacteria
Therapeutic
Antibacterial
Target
GyrB
ParE
Assay information
Inhibitor of DNA gyrase in E. coli (IC50 = 0.5 μM)
Inhibitor of GryB (IC50 = 0.03 μM) and ParE (IC50 = 1.32 μM)
MIC [μg/ml]: S. aureus (0.125), E. faecalis (8), E. coli (8)